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AZ876
CAS No. 898800-26-5
AZ876 ( —— )
产品货号. M19966 CAS No. 898800-26-5
AZ876 is a potent highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥664 | 有现货 |
|
| 10MG | ￥1021 | 有现货 |
|
| 25MG | ￥1337 | 有现货 |
|
| 50MG | ￥1677 | 有现货 |
|
| 100MG | ￥2989 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称AZ876
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述AZ876 is a potent highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.
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产品描述AZ876 is a potent highly selective LXR agonist with Ki/EC50 of 7/6 nM and 11/73 nM for hLXRα and hLXRβ respectively.
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同义词——
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通路Others
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靶点Other Targets
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受体LXR
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研究领域——
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适应症——
化学信息
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CAS Number898800-26-5
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分子量439.57
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分子式C24H29N3O3S
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纯度>98% (HPLC)
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溶解度DMSO: 2.5 mg/mL
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SMILESCC(C)(C)N1C(=O)C(Nc2ccc(cc2)N2CCCCC2)=C(c2ccccc2)S1(=O)=O
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化学全称2-(11-Dimethylethyl)-5-phenyl-4-[[4-(1-piperidinyl)phenyl]amino]-3(2H)-isothiazolone 11-dioxide
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.van der Hoorn J et al. Low dose of the liver X receptor agonist AZ876 reduces atherosclerosis in APOE*3Leiden mice without affecting liver or plasma triglyceride levels. Br J Pharmacol. 2011 Apr;162(7):1553-63.
产品手册
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