
AZ-Dyrk1B-33
CAS No. 1679330-37-0
AZ-Dyrk1B-33 ( 3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine )
产品货号. M26618 CAS No. 1679330-37-0
AZ-Dyrk1B-33 是一种有效的选择性 Dyrk1B 激酶抑制剂,IC50 为 7 nM。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥1320 | 有现货 |
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10MG | ¥2130 | 有现货 |
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25MG | ¥4317 | 有现货 |
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50MG | ¥6278 | 有现货 |
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100MG | ¥8748 | 有现货 |
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500MG | ¥17577 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称AZ-Dyrk1B-33
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述AZ-Dyrk1B-33 是一种有效的选择性 Dyrk1B 激酶抑制剂,IC50 为 7 nM。
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产品描述AZ-Dyrk1B-33 is a potent and selective Dyrk1B kinase inhibitor with an IC50 of 7 nM.(In Vitro):Administration of AZ-Dyrk1B-33 shows inhibition of phosphorylation of Dyrk pS421 in cells with an IC50 of 0.192 μM and no effect in sensitization.
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体外实验AZ-Dyrk1B-33 shows inhibition of phosphorylation of Dyrk pS421 in cells with an IC50 of 0.192 μM.AZ-Dyrk1B-33 shows no effect in sensitization.
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体内实验——
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同义词3-(2-Methyl-4-pyrimidinyl)-1-(phenylmethyl)-1H-pyrrolo[2,3-c]pyridine
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通路Others
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靶点Other Targets
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受体CYP73A
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研究领域——
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适应症——
化学信息
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CAS Number1679330-37-0
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分子量300.365
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分子式C19H16N4
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO : 125 mg/mL (416.17 mM)
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SMILESCc1nccc(n1)-c1cn(Cc2ccccc2)c2cnccc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.1. Schalk M, et al, Werck-Reichhart D. Piperonylic acid, a selective, mechanism-based inactivator of the trans-cinnamate 4-hydroxylase: A new tool to control the flux of metabolites in the phenylpropanoid pathway. Plant Physiol. 1998;118(1):209‐218.
产品手册




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