AGN192836 ( AGN 192836 )

产品货号. M12609 CAS No. 171102-29-7

COA

Datasheet

HNMR

HPLC

MSDS

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产品名称

AGN192836
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

AGN192836 (AGN 192836) is a potent, selective α2 adrenergic (alpha 2-adrenoceptor) agonist with EC50 of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively.
产品描述

AGN192836 (AGN 192836) is a potent, selective α2 adrenergic (alpha 2-adrenoceptor) agonist with EC50 of 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor, respectively; displays 1200-, 50- and 10-fols selectivity for the α2A-receptor, α2B-receptor, and α2C-receptors relative to the α2C-receptors; demonstrates effectivity for the reduction of intraocular pressure and for the reduction of blood pressure in vivo.
同义词

AGN 192836
通路

Angiogenesis
靶点

Adrenergic Receptor
受体

Adrenergic Receptor
研究领域

Cardiovascular Disease
适应症

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1. Munk SA, et al. J Med Chem. 1997 Jan 3;40(1):18-23.

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