A-867744
CAS No. 1000279-69-5
A-867744 ( —— )
产品货号. M23206 CAS No. 1000279-69-5
A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥316 | 有现货 |
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5MG | ¥518 | 有现货 |
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10MG | ¥786 | 有现货 |
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25MG | ¥1563 | 有现货 |
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50MG | ¥2811 | 有现货 |
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100MG | ¥4204 | 有现货 |
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200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
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生物学信息
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产品名称A-867744
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).
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产品描述A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).
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同义词——
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通路Autophagy
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靶点Autophagy
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受体Autophagy;α7 nAChR
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研究领域——
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适应症——
化学信息
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CAS Number1000279-69-5
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分子量402.9
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分子式C20H19ClN2O3S
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纯度>98% (HPLC)
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溶解度DMSO:100 mg/mL (248.21 mM)
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SMILESCCC(c(cc1-c(cc2)ccc2Cl)c(C)n1-c(cc1)ccc1S(N)(=O)=O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Malysz J, et al. In vitro pharmacological characterization of a novel allosteric modulator of alpha 7 neuronal acetylcholine receptor, 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744), exhibiting unique pharmacological profile. J Pharmacol Exp Ther. 2009 Jul;330(1):257-67.
产品手册
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