3-Bromocytisine
CAS No. 207390-14-5
3-Bromocytisine ( 3-Br-cytisine; (-)-3-Bromocytisine; (-)-9-Bromocytisine )
产品货号. M26025 CAS No. 207390-14-5
3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
5MG | ¥1936 | 有现货 |
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10MG | ¥2633 | 有现货 |
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25MG | ¥4439 | 有现货 |
|
50MG | ¥6383 | 有现货 |
|
100MG | ¥8748 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称3-Bromocytisine
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).
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产品描述3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).(In Vitro):3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively .
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同义词3-Br-cytisine; (-)-3-Bromocytisine; (-)-9-Bromocytisine
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通路Others
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靶点Other Targets
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受体D4
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研究领域——
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适应症——
化学信息
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CAS Number207390-14-5
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分子量269.1
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分子式C11H13BrN2O
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纯度>98% (HPLC)
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溶解度——
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SMILESBrc1ccc2[C@H]3CNC[C@H](C3)Cn2c1=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Nakazawa S, et al. Behavioral and neurophysiological effects of Ro 10-5824, a dopamine D4 receptor partial agonist, in common marmosets. Psychopharmacology (Berl). 2015 Sep;232(17):3287-95.
产品手册
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