5-Benzyloxygramine ( —— )

产品货号. M28056 CAS No. 1453-97-0

COA

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HNMR

HPLC

MSDS

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产品名称

5-Benzyloxygramine
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
产品描述

5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.(In Vitro):5-Benzyloxygramine is a new N protein PPI orthosteric stabilizer that exhibits both antiviral and N-NTD protein-stabilizing activities. 5-benzyloxygramine stabilizes the N-NTD dimers through simultaneous hydrophobic interactions with both partners, resulting in abnormal N protein oligomerization that was further confirmed in the cell.
同义词

——
通路

GPCR/G Protein
靶点

Dopamine Receptor
受体

AQP1
研究领域

——
适应症

——

1.Seeliger D, et al. Discovery of novel human aquaporin-1 blockers. ACS Chem Biol. 2013 Jan 18;8(1):249-56.

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